N-Silyl Protecting Groups for Labile Aziridines: Application toward the Synthesis of NH Aziridinomitosenes
DL Warner, AM Hibberd, M Kalman…
Index: Leroy, Jacques; Cantacuzene, Daniele; Wakselman, Claude Synthesis, 1982 , # 4 p. 313 - 315
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Citation Number: 12
Abstract
... In the course of several synthesis projects in our laboratories, we have encountered the need to ... 3, 4, and 5 (isolated yields of 35%, 2 41%, 1 and 65%, 4,5 respectively ... For example, deprotection of aziridinomitosene 2 (PG = trityl) led to the formation of an amorphous precipitate ...
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