Discovery of novel N-phenylphenoxyacetamide derivatives as EthR inhibitors and ethionamide boosters by combining high-throughput screening and synthesis

M Flipo, N Willand, N Lecat-Guillet…

Index: Journal of Medicinal Chemistry, , vol. 55, # 14 p. 6391 - 6402

Full Text: HTML

Citation Number: 17

Abstract

... Journal of Medicinal Chemistry. ... Chem. , 2012, 55 (14), pp 6391–6402. DOI: 10.1021/ jm300377g. Publication Date (Web): June 28, 2012. Copyright © 2012 American Chemical Society. *E-mail: benoit.deprez@univ-lille2.fr. Phone: +33 320 964 947. ...

Related Articles:

Synthesis, structures and the biological activity study on the metal complexes of 2-(4-aminophenyl) benzothiazole derivative

[Lin, Guo-Wu; Wang, Yue; Jin, Qiao-Mei; Yang, Tao-Tao; Song, Jie-Mei; Lu, Yi; Huang, Qing-Jie; Song, Ke; Zhou, Jun; Lu, Tao Inorganica Chimica Acta, 2012 , vol. 382, # 1 p. 35 - 42]

One-step synthesis of 2-arylbenzothiazole ('BTA') and-benzoxazole precursors for in vivo imaging of β-amyloid plaques

[Alagille, David; Baldwin, Ronald M.; Tamagnan, Gilles D. Tetrahedron Letters, 2005 , vol. 46, # 8 p. 1349 - 1351]

An efficient palladium catalyzed synthesis of 2-arylbenzothiazoles

[Majo, Vattoly J.; Prabhakaran, Jaya; Mann, J. John; Kumar, J. S. Dileep Tetrahedron Letters, 2003 , vol. 44, # 47 p. 8535 - 8537]

Antitumor benzothiazoles. 3. 1 Synthesis of 2-(4-aminophenyl) benzothiazoles and evaluation of their activities against breast cancer cell lines in vitro and in vivo

[Journal of Medicinal Chemistry, , vol. 39, # 17 p. 3375 - 3384]

Antitumor benzothiazoles. 3. 1 Synthesis of 2-(4-aminophenyl) benzothiazoles and evaluation of their activities against breast cancer cell lines in vitro and in vivo

[Journal of Medicinal Chemistry, , vol. 39, # 17 p. 3375 - 3384]

More Articles...