Novel imidazobenzazepine derivatives as dual H 1/5-HT 2A antagonists for the treatment of sleep disorders

M Gianotti, C Corti, S Delle Fratte, R Di Fabio…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 20, # 17 p. 5069 - 5073

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Citation Number: 9

Abstract

... Bioorganic & Medicinal Chemistry Letters. ... All the newly prepared chemical entities were assayed for their agonistic and antagonistic properties using two kinds of ... In particular, compounds 19, 20, and 21 were the result of a tailored medicinal chemistry strategy focused on ...

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