Organic letters

β-Aminoethyltrifluoroborates: efficient aminoethylations via Suzuki-Miyaura cross-coupling

GA Molander, F Vargas

Index: Molander, Gary A.; Vargas, Fabricio Organic Letters, 2007 , vol. 9, # 2 p. 203 - 206

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Citation Number: 41

Abstract

A set of phenethylamines has been successfully prepared via Suzuki-Miyaura cross- coupling of diverse potassium β-aminoethyltrifluoroborates with aryl halides. The potassium β-aminoethyltrifluoroborates were easily prepared via hydroboration of enamine and enamide precursors.

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