Synthesis and biological activities of aryl-ether-, biaryl-, and fluorene-aspartic acid and diaminopropionic acid analogs as potent inhibitors of the high-affinity glutamate …

A Greenfield, C Grosanu, J Dunlop, B McIlvain…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 15, # 22 p. 4985 - 4988

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Citation Number: 18

Abstract

... Bioorganic & Medicinal Chemistry Letters. ... In comparison with TBOA series, 7 these inhibitors possess only one chiral center and a free carboxylic acid group, potentially simplifying the syntheses and improving physico-chemical properties. ...