Tetrahedron Letters

A simple acylation of thiols with anhydrides

A Temperini, D Annesi, L Testaferri, M Tiecco

Index: Temperini, Andrea; Annesi, Diego; Testaferri, Lorenzo; Tiecco, Marcello Tetrahedron Letters, 2010 , vol. 51, # 41 p. 5368 - 5371

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Citation Number: 8

Abstract

Download PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... Different thiols were efficiently acylated at room temperature with different anhydrides in the presence of potassium carbonate. Chemoselective protection of thiol in the presence of hydroxy group was achieved using di-tert-butyl dicarbonate and isatoic anhydride.