Intramolecular Cycloisomerization of Aryl-Substituted Alkylidenecyclopropanes via NHC Palladium-Catalyzed Cascade CC Bond Cleavage/CH Activation/CC Bond …
Y Yang, X Huang
Index: Yang, Yewei; Huang, Xian Synlett, 2008 , # 9 p. 1366 - 1370
Full Text: HTML
Citation Number: 0
Abstract
Abstract A well-defined N-heterocyclic carbene (NHC) palladium-catalyzed intramolecular cyclization reaction of aryl-substituted alkylidenecyclopropanes (ACP) to 1-aryl dihydronaphthalenes is described. The NHC salts were found to suppress β-hydride elimination from the homoallylpalladium intermediate, which may lead to unwanted alkene formation. A plausible mechanism for the cycloisomerization was proposed.
Related Articles:
[Hamze, Abdallah; Brion, Jean-Daniel; Alami, Mouad Organic Letters, 2012 , vol. 14, # 11 p. 2782 - 2785]
[Guthrie, Robert W.; Kaplan, Gerald L.; Mennona, Francis A.; Tilley, Jefferson W.; Kierstead, Richard W.; et al. Journal of Medicinal Chemistry, 1990 , vol. 33, # 10 p. 2856 - 2864]
[Guthrie, Robert W.; Kaplan, Gerald L.; Mennona, Francis A.; Tilley, Jefferson W.; Kierstead, Richard W.; et al. Journal of Medicinal Chemistry, 1990 , vol. 33, # 10 p. 2856 - 2864]
[Guthrie, Robert W.; Kaplan, Gerald L.; Mennona, Francis A.; Tilley, Jefferson W.; Kierstead, Richard W.; et al. Journal of Medicinal Chemistry, 1990 , vol. 33, # 10 p. 2856 - 2864]
[Bergmann; Szmuszkowicz; Fawaz Journal of the American Chemical Society, 1947 , vol. 69, p. 1773,1776]