Tetrahedron letters

Traceless solid phase synthesis of 2, 3-disubstituted indoles

AL Smith, GI Stevenson, CJ Swain, JL Castro

Index: Smith, Adrian L.; Stevenson, Graeme I.; Swain, Christopher J.; Castro, Jose L. Tetrahedron Letters, 1998 , vol. 39, # 45 p. 8317 - 8320

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Citation Number: 103

Abstract

Download full text in PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... An efficient method for the traceless solid phase synthesis of 2,3-disubstituted indoles using a THP linker and a Pd(0)-mediated annulation of 2-iodoaniline and acetylenes is reported. ... A THP solid phase linker for indoles, and its use in a Pd(0)-mediated solid phase indole ...

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