A new, general entry to 4-substituted indoles. Synthesis of (S)-(−)-pindolol and (±)-chuangxinmycin

…, T Tabata, K Hanaoka, H Iriyama, S Akamatsu…

Index: Ishibashi, Hiroyuki; Tabata, Takashi; Hanaoka, Kyoko; Iriyama, Hiroko; Akamatsu, Susumu; Ikeda, Masazumi Tetrahedron Letters, 1993 , vol. 34, # 3 p. 489 - 492

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Citation Number: 26

Abstract

Download full text in PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... A new method for synthesis of 4-substituted indoles has been developed by using the 7-arylthio-6-7-dihydroindol-4(5H) one5 as a common intermediate. The method was applied to the synthesis of (S)-(−)-pindolol (11) and (±)-chuangxinmycin (16).