A new synthesis of the GPIIb/IIIa receptor antagonist SB-214857-A

IP Andrews, RJ Atkins, NF Badham, RK Bellingham…

Index: Tetrahedron Letters, , vol. 42, # 29 p. 4915 - 4917

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Citation Number: 27

Abstract

... Tetrahedron Letters. Volume 42, Issue 29, 16 July 2001, Pages 4915–4917. ... In this letter we report an alternative enantioselective synthesis of 1 in which the key intermediate, racemic 1,4-benzodiazepine ester 2, is prepared from 2-nitrobenzyl alcohol 3 using a novel ...

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