Modification and structure–activity relationship of a small molecule HIV-1 inhibitor targeting the viral envelope glycoprotein gp120

J Wang, N Le, A Heredia, H Song, R Redfield…

Index: Organic and Biomolecular Chemistry, , vol. 3, # 9 p. 1781 - 1786

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Citation Number: 40

Abstract

... All reagents were purchased from Aldrich Chemical Co ... 20 mmol) in dry CH 2 Cl 2 (100 ml) under an argon atmosphere at room temperature were added methyl benzoate (2.72 g, 2.5 ml, 20 mmol) and Et 2 AlCl 3 (1.0 M ... The organic layer was dried over MgSO 4 and concentrated ...

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