Cardioselective antiischemic ATP-sensitive potassium channel openers. 2. structure-activity studies on benzopyranylcyanoguanidines; modification of the benzopyran …
…, GJ Grover, FN Ferrara, SZ Ahmed…
Index: Atwal, Karnail S.; Grover, Gary J.; Ferrara, Francis N.; Ahmed, Syed Z.; Sleph, Paul G.; et al. Journal of Medicinal Chemistry, 1995 , vol. 38, # 11 p. 1966 - 1973
Full Text: HTML
Citation Number: 59
Abstract
The ATP-sensitive potassium channel (KATP) openers are of considerable interest as myocardial protecting agents. However, there exists a narrow window of safety for the use of firstgeneration compounds as antiischemic agents due to their powerful peripheral vasodilating effects, which can result in underperfusion of the area already at risk. We have recently disclosed the discovery of benzopyranylcyanoguanidine type KATP openers ( ...
Related Articles:
[Tsuzuki, Yasuhiro; Nguyen, Thao Kim Nu; Garud, Dinesh R.; Kuberan, Balagurunathan; Koketsu, Mamoru Bioorganic and Medicinal Chemistry Letters, 2010 , vol. 20, # 24 p. 7269 - 7273]
[Gonzalez-Gomez, Alvaro; Anorbe, Loreto; Poblador, Amalia; Dominguez, Gema; Perez-Castells, Javier European Journal of Organic Chemistry, 2008 , # 8 p. 1370 - 1377]
[Chaudhuri, Subrata Kumar; Roy, Sanchita; Saha, Manabendra; Bhar, Sanjay Synthetic Communications, 2007 , vol. 37, # 2 p. 271 - 274]
[Powell; Adams Journal of the American Chemical Society, 1920 , vol. 42, p. 655]
[Powell; Adams Journal of the American Chemical Society, 1920 , vol. 42, p. 655]