Organic Letters

Diastereoselectively Complementary C–H Functionalization Enables Access to Structurally and Stereochemically Diverse 2, 6-Substituted Piperidines

G Wang, Y Mao, L Liu

Index: Barbe, Guillaume; St-Onge, Miguel; Charette, Andre B. Organic Letters, 2008 , vol. 10, # 23 p. 5497 - 5499

Full Text: HTML

Citation Number: 1

Abstract

... Organic Letters. Advanced Search. ... Table 1. Reaction Condition Optimization a. entry, oxidant, yield (%) b of 3a/3″a, dr c. 1 d, oxidant, <5, na. 2, TEMPO + OTf –, 50/25, 7:1. 3, TEMPO + ClO 4 –, 66/12, 10:1. 4, TEMPO + BF 4 –, 76/<5, 12:1. 5 e, TEMPO + BF 4 –, 73/13, 16:1. ...

Related Articles:

Synthesis of diastereomerically and enantiomerically pure 2, 3-disubstituted tetrahydrofurans using a sulfoxonium ylide

[Schomaker, Jennifer M.; Pulgam, Veera Reddy; Borhan, Babak Journal of the American Chemical Society, 2004 , vol. 126, # 42 p. 13600 - 13601]

A novel nonpeptide HIV-1 protease inhibitor: elucidation of the binding mode and its application in the design of related analogs

[Lunney; Hagen; Domagala; Humblet; Kosinski; Tait; Warmus; Wilson; Ferguson; Hupe; Tummino; Baldwin; Bhat; Liu; Erickson Journal of Medicinal Chemistry, 1994 , vol. 37, # 17 p. 2664 - 2677]

Synthesis and structure-activity relationships of soluble 7-substituted 3-(3, 5-dimethoxyphenyl)-1, 6-naphthyridin-2-amines and related ureas as dual inhibitors of the …

[Thompson, Andrew M.; Delaney, Amy M.; Hamby, James M.; Schroeder, Mel C.; Spoon, Teresa A.; Crean, Sheila M.; Showalter, H. D. Hollis; Denny, William A. Journal of Medicinal Chemistry, 2005 , vol. 48, # 14 p. 4628 - 4653]

Synthesis of novel spiro heterocycles. 2-Amino-7-oxa-3-thia-1-azaspiro [5.5] undec-1-enes

[Cohen,N. et al. Journal of Organic Chemistry, 1974 , vol. 39, p. 1824 - 1833]

1, 2-Silyl-Migrative Cyclization of Vinylsilanes Bearing a Hydroxy Group: Stereoselective Synthesis of Multisubstituted Tetrahydropyrans and Tetrahydrofurans1

[Miura, Katsukiyo; Hondo, Takeshi; Okajima, Shigeo; Nakagawa, Takahiro; Takahashi, Tatsuyuki; Hosomi, Akira Journal of Organic Chemistry, 2002 , vol. 67, # 17 p. 6082 - 6090]

More Articles...