Tetrahedron Letters

Acetals: a new organocatalysis chemotype for one-pot enantioselective α-amination

R Hunter

Index: Msutu, Ath'Enkosi; Hunter, Roger Tetrahedron Letters, 2014 , vol. 55, # 14 p. 2295 - 2298

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Citation Number: 6

Abstract

Abstract Conditions are described for one-pot Brønsted acid and organocatalysed enantioselective α-amination of acetals and associated functionalities. Of the organocatalysts screened, proline tetrazole gave the highest ee, while aqueous ...