New proline mimetics: synthesis of thrombin inhibitors incorporating cyclopentane-and cyclopentenedicarboxylic acid templates in the P2 position. Binding …

D Nöteberg, J Brånalt, I Kvarnström…

Index: Lila, Christine; Gloanec, Philippe; Cadet, Laurence; Herve, Yolande; Fournier, Jean; Leborgne, Fabrice; Verbeuren, Tony J.; De Nanteuil, Guillaume Synthetic Communications, 1998 , vol. 28, # 23 p. 4419 - 4429

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Citation Number: 38

Abstract

... Volume: Page: ... J. Med. Chem. ... Numerous synthetic routes for the desired enantiomerically pure trans-cyclopentane-1,2-dicarboxylic acid derivatives have been reported, including traditional resolution, 11 enzymatic resolution, 12 and asymmetric synthesis. ...

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