Discovery of potent and selective nonsteroidal indazolyl amide glucocorticoid receptor agonists
JE Sheppeck, JL Gilmore, HY Xiao, TGM Dhar…
Index: Bioorganic and Medicinal Chemistry Letters, , vol. 23, # 19 p. 5442 - 5447
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Citation Number: 7
Abstract
... Bioorganic & Medicinal Chemistry Letters. ... The indazoles in this and the accompanying Letter were all synthesized from the common synthetic intermediate 5- hydroxymethylindazole (Scheme 1) prepared using the method of Sun et al. ...
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