ChemMedChem

Design and synthesis of tricyclic JAK3 inhibitors with picomolar affinities as novel molecular probes

M Gehringer, E Pfaffenrot, S Bauer…

Index: ChemMedChem, , vol. 9, # 2 p. 277 - 281

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Citation Number: 12

Abstract

... Probes. ChemMedChem, 9: 277–281. doi: 10.1002/cmdc.201300520. Author Information. ... SEARCH BY CITATION. Volume: Issue: Page: ... geometry. Finally, benzylated precursor 9 showed poor inhibitory activity in the low micromolar range. ...