Tetrahedron Letters

Synthèse D'α, β-fluoroamines à partir d'aziridines: orientation de l'ouverture du cycle et amélioration du pouvoir fluorant du réactif de olah

G Alvernhe, S Lacombe, A Laurent

Index: Alvernhe, Gerard; Lacombe, Sylvie; Laurent, Andre Tetrahedron Letters, 1980 , vol. 21, p. 289 - 292

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Citation Number: 26

Abstract

Résumé Ring opening of aliphatic and aromatic aziridines by addition of Olah's reagent has been studied. Yields and regioselectivity are improved when using the corresponding N- activated aziridines and less acidic fluorinating reagents obtained by addition of triethylamine to Olah's reagent.

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