Tetrahedron Letters

Inverse electron-demand Diels–Alder chemistry in the synthesis of a regioselectively protected analogue of the staurosporine aglycone

R Nomak, JK Snyder

Index: Nomak, Rana; Snyder, John K. Tetrahedron Letters, 2001 , vol. 42, # 45 p. 7929 - 7933

Full Text: HTML

Citation Number: 32

Abstract

Regioselective Weinreb amidation of the C1 ester of dimethyl pyridazino [4, 5-b] indole-1, 4- dicarboxylate followed by an intramolecular inverse electron-demand Diels–Alder reaction and palladium-catalyzed coupling produced regioselectively protected N6-methylindolo [2, 3- a] pyrrolo [3, 4-c] carbazole (N6-methylstaurosporinone).

Related Articles:

Highly selective TFAA-cleavage of tertiary 2, 4-dimethoxybenzylamines and its use in the synthesis of secondary amines

[Nussbaumer; Baumann; Dechat; Harasek Tetrahedron, 1991 , vol. 47, # 26 p. 4591 - 4602]

Mild and efficient synthesis of propargylamines by copper-catalyzed Mannich reaction

[Bieber, Lothar W.; Da Silva, Margarete F. Tetrahedron Letters, 2004 , vol. 45, # 45 p. 8281 - 8283]

Cationic dirhodium carboxylate-catalyzed synthesis of dihydropyrimidones from propargyl ureas

[Yang, Miao; Odelberg, Shannon J.; Tong, Zongzhong; Li, Dean Y.; Looper, Ryan E. Tetrahedron, 2013 , vol. 69, # 27-28 p. 5744 - 5750]

Cationic dirhodium carboxylate-catalyzed synthesis of dihydropyrimidones from propargyl ureas

[Yang, Miao; Odelberg, Shannon J.; Tong, Zongzhong; Li, Dean Y.; Looper, Ryan E. Tetrahedron, 2013 , vol. 69, # 27-28 p. 5744 - 5750]

More Articles...