2-Substituted 5-methoxy-N-acyltryptamines: synthesis, binding affinity for the melatonin receptor, and evaluation of the biological activity

G Spadoni, B Stankov, A Duranti, G Biella…

Index: Journal of Medicinal Chemistry, , vol. 36, # 25 p. 4069 - 4074

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Citation Number: 78

Abstract

... 0022-2623/93/1836-4069$04.00/0 @ 1993 American Chemical Society Page 2. 4070 Journal of Medicinal Chemistry, 1993, Vol. 36, No. 25 Spadoni et al. 5.8 X for 2-bromomelatonin) decrease in the apparent binding affinity of the new compound. ...

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