Tetrahedron letters

A new approach to the synthesis of lavendamycin analogues.

P Rocca, F Marsais, A Godard, G Quéguiner

Index: Rocca, Patrick; Marsais, Fracis; Godard, Alain; Queguiner, Guy Tetrahedron Letters, 1993 , vol. 34, # 18 p. 2937 - 2940

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Citation Number: 37

Abstract

Abstract A three-steps approach to the lavendamycin skeleton from benzene, pyridine and quinoline blocks is described. It is based on a new synthetic methodology for the preparation of α-substituted β-carbolines which involves such reactions as Directed Ortho Metalation and Heteroring Cross-Coupling.

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