An efficient synthesis of N-benzyl-3-sulfonyl glutarimides. Formal synthesis of the aromatase inhibitor AG-1
MY Chang, BR Chang, HM Tai, NC Chang
Index: Chang, Meng-Yang; Chang, Bo-Rui; Tai, Huo-Mu; Chang, Nein-Chen Tetrahedron Letters, 2000 , vol. 41, # 52 p. 10273 - 10276
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Abstract
Download PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... A formal [3+3] cycloaddition strategy to substituted glutarimides was studied. N-Benzyl α-sulfonylacetamides and various α,β-unsaturated esters were used as starting materials. ... Sequential treatment of chloroacetyl chloride with benzylamine and sodium p-toluenesulfinate furnished α- ...
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