Tetrahedron Letters

Solvent-free Mukaiyama and Mukaiyama–Michael vinylogous reactions of a dioxinone-derived silyl enol ether promoted by Lewis bases

A Scettri, V De Sio, R Villano, P Manzo, MR Acocella

Index: Scettri, Arrigo; Sio, Vincenzo De; Villano, Rosaria; Manzo, Patrizia; Acocella, Maria Rosaria Tetrahedron Letters, 2010 , vol. 51, # 28 p. 3658 - 3661

Full Text: HTML

Citation Number: 8

Abstract

The vinylogous aldol-type addition of a dienolsilyl ether, derived from 2, 2, 6-trimethyl-4H-1, 3-dioxin-4-one, showed to occur with complete γ-selectivity by enolate activation promoted by neutral Lewis bases under solvent-free conditions. Moderate to high yields were obtained with aromatic, hetero-aromatic, and aliphatic aldehydes, as well as activated ketones. Under the same conditions and in the absence of catalyst, the first Mukaiyama–Michael addition ...

Related Articles:

Stereoselective synthesis of tetrahydropyran-4-ones from dioxinones catalyzed by scandium (III) triflate

[Morris, William J.; Custar, Daniel W.; Scheidt, Karl A. Organic Letters, 2005 , vol. 7, # 6 p. 1113 - 1116]

Solvent-free Mukaiyama aldol reaction of O-silyl dienolates catalyzed by benzoic acid

[Acocella, Maria Rosaria; Massa, Antonio; Palombi, Laura; Villano, Rosaria; Scettri, Arrigo Tetrahedron Letters, 2005 , vol. 46, # 36 p. 6141 - 6144]

Solvent-free Mukaiyama aldol reaction of O-silyl dienolates catalyzed by benzoic acid

[Acocella, Maria Rosaria; Massa, Antonio; Palombi, Laura; Villano, Rosaria; Scettri, Arrigo Tetrahedron Letters, 2005 , vol. 46, # 36 p. 6141 - 6144]

More Articles...