Fluorescent non-imidazole histamine H 3 receptor ligands with nanomolar affinities

M Amon, X Ligneau, JC Schwartz, H Stark

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 16, # 7 p. 1938 - 1940

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Citation Number: 18

Abstract

... Bioorganic & Medicinal Chemistry Letters. ... Keywords. Histamine; Antagonist; Ligand; Fluorescence; H3; Medicinal chemistry. ... 16. b The n-octanol/water partition coefficient based on established chemical interactions; calculated with ChemDraw Ultra 7.0. 17. e Value from Ref. 5. ...