Tetrahedron Letters

Copper-catalyzed multicomponent reactions of 2-iodoanilines, benzylamines, and elemental sulfur toward 2-arylbenzothiazoles

R Wang, Y Ding, H Liu, S Peng, J Ren, L Li

Index: Wang, Rui; Ding, Yong-Liang; Liu, Hong; Peng, Shu; Ren, Jie; Li, Lei Tetrahedron Letters, 2014 , vol. 55, # 4 p. 945 - 949

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Citation Number: 4

Abstract

Abstract A relatively cheap copper salt-catalyzed, three-component approach providing 2- arylbenzothiazoles in good to excellent yields from readily available 2-iodoanilines, benzylamines, and sulfur powder is reported. This methodology allows preparation of various classes of 2-arylbenzothiazoles and provides a general, reliable approach.

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