Acidic and basic deprotection strategies of borane-protected phosphinothioesters for the traceless Staudinger ligation

M Mühlberg, J Da'san MM, R Kleineweischede…

Index: Bioorganic and Medicinal Chemistry, , vol. 18, # 11 p. 3679 - 3686

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Citation Number: 10

Abstract

... Bioorganic & Medicinal Chemistry. ... Borane-deprotection under basic conditions for 7a and in situ formation of 10: Temperature measurements after 1 h unless stated otherwise (r = ratio of deprotection/protection according to –SCH 2 P– chemical shifts; '—' = no deprotection ...