Thioperamide (maleate)

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Names

[ Name ]:
Thioperamide (maleate)

[Synonym ]:
MR-12842 N-Cyclohexyl-4-(1H-imidazol-4-yl)-1-piperidinecarbothioamide maleate salt
1-Piperidinecarbothioamide, N-cyclohexyl-4-(1H-imidazol-5-yl)-, (2Z)-2-butenedioate (1:1)
MR-12842 (N-Cyclohexyl-4-(1H-imidazol-4-yl)-1-piperidinecarbothioamide maleate salt
Thioperamide Maleate
N-Cyclohexyl-4-(1H-imidazol-5-yl)-1-piperidinecarbothioamide (2Z)-2-butenedioate (1:1)
1-Piperidinecarbothioamide, N-cyclohexyl-4-(1H-imidazol-4-yl)-, (2Z)-2-butenedioate (1:1)
MFCD00083209
N-Cyclohexyl-4-(1H-imidazol-4-yl)piperidine-1-carbothioamide (2Z)-but-2-enedioate (1:1)

Chemical & Physical Properties

[ Molecular Formula ]:
C₁₉H₂₈N₄O₄S

[ Molecular Weight ]:
408.515

[ Exact Mass ]:
408.183136

[ PSA ]:
150.64000

[ LogP ]:
2.83690

MSDS

Click to get detail MSDS

Safety Information

[ Symbol ]:

GHS07

[ Signal Word ]:
Warning

[ Hazard Statements ]:
H315-H319-H335

[ Precautionary Statements ]:
P261-P305 + P351 + P338

[ Personal Protective Equipment ]:
dust mask type N95 (US);Eyeshields;Gloves

[ Hazard Codes ]:
Xi

[ Risk Phrases ]:
R36/37/38

[ Safety Phrases ]:
S26

[ RIDADR ]:
NONH for all modes of transport

Articles

Highly potent and selective ligands for histamine H3-receptors.

Nature 327 , 117, (1987)

New drugs selective for histamine H3-receptors can be used to establish that these receptors are involved in the feedback control of histamine synthesis and release, and to demonstrate their distribut...

Effects of the histamine H3-agonist (R)-alpha-methylhistamine and the antagonist thioperamide on histamine metabolism in the mouse and rat brain.

J. Neurochem. 52 , 1388, (1989)

To study the feedback control by histamine (HA) H3-receptors on the synthesis and release of HA at nerve endings in the brain, the effects of a potent and selective H3-agonist, (R)-alpha-methylhistami...

Effect of thioperamide, a histamine H3 receptor antagonist, on electrically induced convulsions in mice.

Eur. J. Pharmacol. 234(1) , 129-33, (1993)

The effect of thioperamide, a histamine H3 receptor antagonist, on electrically induced convulsions was studied in mice. Thioperamide significantly and dose dependently decreased the duration of each ...

Thioperamide
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3-[(2-chlorophenyl)methyl]-4-methyl-5aH-pyrimido[1,2-a]benzimidazol-2-one
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N-(4-chlorophenyl)-1,3-dimethyl-2,4,7-trioxo-6H-pyrido[2,3-d]pyrimidin-8-ium-5-carboxamide
2-amino-5-(1,3-benzodioxol-5-yl)-8,8-dimethyl-2,3,4a,5,7,9,10,10a-octahydro-1H-pyrimido[4,5-b]quinoline-4,6-dione
2-[[1-(4-Chlorophenyl)tetrazol-5-yl]methylsulfanyl]-6-methyl-1,3-diazinan-4-one
3-[(1,3-benzodioxol-5-ylmethylamino)methyl]-6-ethoxy-3,4,4a,5,6,7,8,8a-octahydro-1H-quinolin-2-one
ethyl 5,6-dimethyl-4-oxo-4aH-thieno[2,3-d]pyrimidine-2-carboxylate
2-(2-Ethoxyethyl)-4-methyl-6-(4-methylphenyl)-4a,7,8,9a-tetrahydropurino[7,8-a]imidazole-1,3-dione
ethyl 1-[3-(2,4-dioxo-4aH-quinazolin-3-yl)propanoyl]piperidine-4-carboxylate
6-morpholin-4-yl-3-(3-piperidin-1-ylpropyl)-2-sulfanylidene-6H-quinazolin-4-one

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