voxilaprevir

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Names

[ CAS No. ]:
1535212-07-7

[ Name ]:
voxilaprevir

[Synonym ]:
voxilaprevir
GS-9857
(1R,18R,20R,24S,27S,28S)-N-[(1R,2R)-2-(Difluoromethyl)-1-{[(1-methylcyclopropyl)sulfonyl]carbamoyl}cyclopropyl]-28-ethyl-13,13-difluoro-7-methoxy-24-(2-methyl-2-propanyl)-22,25-dioxo-2,21-dioxa-4,11,2 ;3,26-tetraazapentacyclo[24.2.1.0.0.0]nonacosa-3(12),4,6,8,10-pentaene-27-carboxamide
8H-7,10-Methanocyclopropa[18,19][1,10,3,6]dioxadiazacyclononadecino[11,12-b]quinoxaline-8-carboxamide, N-[(1R,2R)-2-(difluoromethyl)-1-[[[(1-methylcyclopropyl)sulfonyl]amino]carbonyl]cyclopropyl]-5-(1,1-dimethylethyl)-9-ethyl-18,18-difluoro-1,1a,3,4,5,6,9,10,18,19,20,21,22,22a-tetradecahydro-14-methoxy-3,6-dioxo-, (1aR,5S,8S,9S,10R,22aR)-
UNII:0570F37359
voxilaprevirum
(1aR,5S,8S,9S,10R,22aR)-5-tert-butyl-N-[(1 R,2R)-2-(difluoromethyl)-1-{[(1-methylcyclopropyl)sulfonyl]carbamoyl}cyclopropyl]-9-ethyl-18,18-difluoro-14- methoxy-3,6-dioxo-1,1a,3,4,5,6,9,1 0,18,19,20,21,22,22a-tetradecahydro-8H-7,10-methanocyclopropa[18,19][1,10,3,6]dioxadiazacyclononadecino[11,12-b]quinoxaline-8-carboxamide
(1aR,5S,8S,9S,10R,22aR)-5-tert-butyl-N-[(1R,2R)-2-(difluoromethyl)-1-{[(1-methylcyclopropyl)sulfonyl]carbamoyl}cyclopropyl]-9-ethyl-18,18-difluoro-14-methoxy-3,6-dioxo-1,1a,3,4,5,6,9,10,18,19,20,21,22,22a-tetradecahydro-8H-7,10-methanocyclopropa[18,19][1,10,3,6]dioxadiazacyclononadecino[11,12-b]quinoxaline-8-carboxamide

Chemical & Physical Properties

[ Density]:
1.4±0.1 g/cm3

[ Molecular Formula ]:
C40H52F4N6O9S

[ Molecular Weight ]:
868.93400

[ Exact Mass ]:
868.34500

[ PSA ]:
203.60000

[ LogP ]:
3.83

[ Index of Refraction ]:
1.596

[ Storage condition ]:
2-8°C

[ Water Solubility ]:
Insuluble (2.8E-4 g/L) (25 ºC)


Related Compounds

  • Voxilaprevir intermediate4
  • Voxilaprevir intermediate1
  • GS9857 (Voxilaprevir) Intermediates
  • 1-methyl-5-(2-methylpyridin-4-yl)-1H-pyrazole-4-carboxylic acid
  • 5-(2-cyclopropylphenyl)-1H-pyrazole-3-carboxylic acid
  • 2-Methyl-2-[6-(pyrrolidin-1-yl)pyridin-3-yl]propanoic acid
  • 2-Hydroxy-2-methyl-3-[2-(propan-2-yl)-1,3-thiazol-4-yl]propanoic acid
  • 3-{Bicyclo[2.2.1]heptan-2-yl}-2-methoxy-3-methylbutanoic acid
  • 2-[1-(3,5-Difluoropyridin-4-yl)cyclobutyl]acetic acid
  • 1-[(4-fluoro-1H-indol-3-yl)methyl]cyclopropane-1-carboxylic acid
  • 2-[4-(Dimethylcarbamoyl)phenyl]propanoic acid
  • rac-(1R,3R)-2,2-dimethyl-3-(quinolin-4-yl)cyclopropane-1-carboxylic acid
  • 3-[2-(Dimethylamino)-4-fluorophenyl]-3-hydroxypropanoic acid