3-Pyridylboronic acid

Suppliers

Names

[ CAS No. ]:
1692-25-7

[ Name ]:
3-Pyridylboronic acid

[Synonym ]:
Acide pyridin-3-ylboronique
3-Pyridineboronic acid
Pyridin-3-bronic Acid
3-Pridylboronic acid
pyridin-3-yl boronic acid
3-Pyridylboronic aci
3-Pyridinylboronic acid
Boronic acid, B-3-pyridinyl-
pyridin-3-ylboronic acid
RARECHEM AH PB 0251
IFLAB-BB F1957-0039
3-pyridineboric acid
Pyridine-3-boronic Acid
3-Pyridylboronic acid
Pyridine-3-acid
MFCD00674177
3-PYRIDINEBORNIC ACID
3-pyridyl boronic acid

Chemical & Physical Properties

[ Density]:
1.2±0.1 g/cm3

[ Boiling Point ]:
308.8±34.0 °C at 760 mmHg

[ Melting Point ]:
>300 °C(lit.)

[ Molecular Formula ]:
C5H6BNO2

[ Molecular Weight ]:
122.92

[ Flash Point ]:
140.5±25.7 °C

[ Exact Mass ]:
123.049156

[ PSA ]:
53.35000

[ LogP ]:
0.10

[ Vapour Pressure ]:
0.0±0.7 mmHg at 25°C

[ Index of Refraction ]:
1.534

[ Storage condition ]:
0-6°C

MSDS

Click to get detail MSDS

Safety Information

[ Personal Protective Equipment ]:
Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter

[ Hazard Codes ]:
Xn:Harmful

[ Risk Phrases ]:
R22;R36/37/38

[ Safety Phrases ]:
S36/37/39-S3-S26

[ RIDADR ]:
NONH for all modes of transport

[ WGK Germany ]:
3

[ HS Code ]:
2933399090

Synthetic Route

Click to get detail synthetic route

Precursor & DownStream

Precursor

  • 3-Bromopyridine
  • Triisopropylborate
  • Trimethyl borate
  • n-Butyllithium
  • Ethanol
  • Tert-Butyllithium
  • Lithium methoxide
  • 4'-Brom-2,2':6',2''-terpyridin
  • 5,5,5',5'-Tetramethyl-2,2'-bi(1,3,2-dioxaborinane)
  • Hydrochloric acid

DownStream

  • 3-azidopyridine
  • 3-Fluoropyridine
  • Phenyl(3-pyridinyl)methanone
  • Latrepirdine
  • 3-(3-Nitrophenyl)pyridine
  • 3-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine
  • 4-Chloromethyl-n-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide
  • 3-trifluoromethylpyridine
  • 3-(5-Imidazolyl)pyridine
  • 3-(3-Methoxyphenyl)pyridine

Customs

[ HS Code ]: 2933399090

[ Summary ]:
2933399090. other compounds containing an unfused pyridine ring (whether or not hydrogenated) in the structure. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:20.0%

Articles

A new access to 3-substituted-1(2H)-isoquinolone by tandem palladium-catalyzed intramolecular aminocarbonylation annulation.

Org. Biomol. Chem. 13th ed., 10 , 2683-2691, (2012)

An original tribromide derivative based, palladium-catalyzed synthesis of 3-substituted-1(2H)-isoquinolone is described based on a regioselective Suzuki-Miyaura C-C coupling on o-halo-(2,2-dihalovinyl...

Synthesis and biological evaluation of novel amprenavir-based P1-substituted bi-aryl derivatives as ultra-potent HIV-1 protease inhibitors.

Bioorg. Med. Chem. Lett. 5th ed., 22 , 1976-1979, (2012)

A series of P1-substituted biaryl amprenavir derivatives was designed and synthesized. These compounds were evaluated for enzyme inhibition and antiviral activity in vitro. Several compounds showed hi...

Copper-mediated sequential cyanation of aryl C-B and arene C-H bonds using ammonium iodide and DMF.

J. Am. Chem. Soc. 5th ed., 134 , 2528-2531, (2012)

The cyanation of aromatic boronic acids, boronate esters, and borate salts was developed under copper-mediated oxidative conditions using ammonium iodide and DMF as the source of nitrogen and carbon a...


More Articles

Related Compounds

  • 4-cyano-3-pyridylboronic acid
  • 4-cyano-3-pyridylboronic acid
  • 2-bromo-3-pyridylboronic acid
  • 4-chloro3-pyridylboronic acid
  • 6-Bromo-3-pyridylboronic Acid
  • 2-cyano-3-pyridylboronic acid
  • N-methyl-N-[1-(pyrazin-2-yl)azetidin-3-yl]-4-(trifluoromethyl)-1,3-benzothiazol-2-amine
  • 4-(3,5-Dimethylpyrazol-1-yl)-6-[4-(2,6-dimethylpyrimidin-4-yl)piperazin-1-yl]-2-methylpyrimidine
  • 2-{4-[(7-Fluoro-2-methyl-4-oxo-3,4-dihydroquinazolin-3-yl)methyl]piperidin-1-yl}pyridine-3-carbonitrile
  • 3-methyl-6-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-[1,2,4]triazolo[4,3-b]pyridazine
  • 6-{4-[(7-Fluoro-2-methyl-4-oxo-3,4-dihydroquinazolin-3-yl)methyl]piperidin-1-yl}pyridine-3-carbonitrile
  • 4-[(1H-imidazol-1-yl)methyl]-N-methyl-N-[1-(pyridin-2-yl)azetidin-3-yl]benzamide
  • 2-Methyl-5-[4-(6-pyrazol-1-ylpyridazin-3-yl)piperazin-1-yl]-1,3,4-thiadiazole
  • 7-Fluoro-3-[[1-(2-pyrazol-1-ylethyl)piperidin-4-yl]methyl]quinazolin-4-one
  • 7-Fluoro-3-[[1-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidin-4-yl]methyl]quinazolin-4-one
  • N-[(1-Thiophen-3-ylcyclopropyl)methyl]-2,3-dihydro-1-benzofuran-5-sulfonamide
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