Norgestimate

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Names

[ CAS No. ]:
35189-28-7

[ Name ]:
Norgestimate

[Synonym ]:
(3E,8R,9S,10R,13S,14S,17R)-13-Ethyl-17-ethynyl-3-(hydroxyimino)-2,3,6,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-17-yl acetate
(+)-13-Ethyl-17-hydroxy-18,19-dinor-17a-pregn-4-en-20-yn-3-one Oxime Acetate (Ester)
d-17beta-acetoxy-13beta-ethyl-17alpha-ethinyl-gon-4en-3-one oxime
dexnorgestrelacetime
Norgestimat
Norgestimate
NORGESTIMATE,USP STANDARD
levonorgestrel acetate 3-oxime
(3E,8R,9S,10R,13S,14S,17R)-17-Ethinyl-13-ethyl-3-(hydroxyimino)-2,3,6,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-17-ylacetat
acétate de (3E,8R,9S,10R,13S,14S,17R)-13-éthyl-17-éthynyl-3-(hydroxyimino)-2,3,6,7,8,9,10,11,12,13,14,15,16,17-tétradécahydro-1H-cyclopenta[a]phénanthrén-17-yle

Chemical & Physical Properties

[ Density]:
1.2±0.1 g/cm3

[ Boiling Point ]:
497.9±45.0 °C at 760 mmHg

[ Melting Point ]:
216ºC

[ Molecular Formula ]:
C23H31NO3

[ Molecular Weight ]:
369.497

[ Flash Point ]:
254.9±28.7 °C

[ Exact Mass ]:
369.230408

[ PSA ]:
58.89000

[ LogP ]:
5.00

[ Vapour Pressure ]:
0.0±2.9 mmHg at 25°C

[ Index of Refraction ]:
1.611

MSDS

Toxicological Information

CHEMICAL IDENTIFICATION

RTECS NUMBER :
JF7976000
CHEMICAL NAME :
18,19-Dinorpregn-4-en-20-yn-3-one, 17-(acetyloxy)-13-ethyl-, 3-oxime, (17-alpha)-
CAS REGISTRY NUMBER :
35189-28-7
LAST UPDATED :
198910
DATA ITEMS CITED :
1
MOLECULAR FORMULA :
C23-H31-N-O3
MOLECULAR WEIGHT :
369.55

HEALTH HAZARD DATA

ACUTE TOXICITY DATA

TYPE OF TEST :
TDLo - Lowest published toxic dose
ROUTE OF EXPOSURE :
Oral
DOSE :
1 mg/kg
SEX/DURATION :
female 2 day(s) pre-mating
TOXIC EFFECTS :
Reproductive - Fertility - other measures of fertility
REFERENCE :
CCPTAY Contraception. (Geron-X, Inc., POB 1108, Los Altos, CA 94022) V.1- 1970- Volume(issue)/page/year: 16,541,1977

Safety Information

[ Symbol ]:

GHS07, GHS08

[ Signal Word ]:
Warning

[ Hazard Statements ]:
H302-H315-H319-H361fd

[ Precautionary Statements ]:
P281-P305 + P351 + P338

[ Hazard Codes ]:
Xn

[ Risk Phrases ]:
63-22-36/38-62

[ Safety Phrases ]:
26-36/37

[ RIDADR ]:
NONH for all modes of transport

[ RTECS ]:
JF7976000

Synthetic Route

Precursor & DownStream

Precursor

  • (8R,9S,10R,13S,14S,17R)-13-Ethyl-17-ethynyl-3-oxo-2,3,6,7,8,9,10, 11,12,13,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-1 7-yl acetate (non-preferred name)

DownStream

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