10,11-Dihydrocarbamazepine

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Names

[ CAS No. ]:
3564-73-6

[ Name ]:
10,11-Dihydrocarbamazepine

[Synonym ]:
10,11-dihydro-5-carboxamido-5H-dibenz<b,f>azepine
10,11-Dihydro-5-carbamoyl-5H-dibenz<b,f>azepin
10,11-Dihydro-5-carbamoyl-5H-dibenz<b,f>azepine
GP 26-301
10,11-DIHYDROCARBAMAZEPINE
EINECS 222-649-0
10,11-Dihydro-5H-dibenz[b,f]azepine-5-carboxamide
10,11-Dihydrocarbamazepine,10,11-Dihydro-5H-dibenz[b,f]azepine-5-carboxamide
MFCD00005072
10,11-Dihydro-5H-dibenz(b,f)azepine-5-carboxamide
10,11-Dihydro-5H-dibenzo[b,f]azepine-5-carboxamide
5H-DIBENZ(b,f)AZEPINE-5-CARBOXAMIDE,10,11-DIHYDRO
5H-Dibenz[b,f]azepine-5-carboxamide, 10,11-dihydro-

Chemical & Physical Properties

[ Density]:
1.2±0.1 g/cm3

[ Boiling Point ]:
394.5±52.0 °C at 760 mmHg

[ Melting Point ]:
205-210ºC

[ Molecular Formula ]:
C15H14N2O

[ Molecular Weight ]:
238.28

[ Flash Point ]:
192.4±30.7 °C

[ Exact Mass ]:
238.110611

[ PSA ]:
46.33000

[ LogP ]:
2.60

[ Vapour Pressure ]:
0.0±0.9 mmHg at 25°C

[ Index of Refraction ]:
1.645

[ Storage condition ]:
Refrigerator

[ Water Solubility ]:
dichloromethane: soluble2.5%, clear, colorless | Soluble in dichloromethane. Insoluble in water.

MSDS

Toxicological Information

CHEMICAL IDENTIFICATION

RTECS NUMBER :
HN8300000
CHEMICAL NAME :
5H-Dibenz(b,f)azepine-5-carboxamide, 10,11-dihydro-
CAS REGISTRY NUMBER :
3564-73-6
BEILSTEIN REFERENCE NO. :
0196969
LAST UPDATED :
199712
DATA ITEMS CITED :
1
MOLECULAR FORMULA :
C15-H14-N2-O
MOLECULAR WEIGHT :
238.31
WISWESSER LINE NOTATION :
T C676 BN&T&J BVZ

HEALTH HAZARD DATA

ACUTE TOXICITY DATA

TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Intraperitoneal
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
750 mg/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
JMCMAR Journal of Medicinal Chemistry. (American Chemical Soc., Distribution Office Dept. 223, POB POB 57136, West End Stn., Washington, DC 20037) V.6- 1963- Volume(issue)/page/year: 7,88,1964

Safety Information

[ Symbol ]:

GHS07, GHS08

[ Signal Word ]:
Danger

[ Hazard Statements ]:
H302-H317-H334

[ Precautionary Statements ]:
P261-P280-P342 + P311

[ Hazard Codes ]:
Xn

[ Risk Phrases ]:
22-42/43

[ Safety Phrases ]:
S24/25

[ RIDADR ]:
NONH for all modes of transport

[ WGK Germany ]:
3

[ RTECS ]:
HN8300000

[ HS Code ]:
2933990090

Synthetic Route

Customs

[ HS Code ]: 2933990090

[ Summary ]:
2933990090. heterocyclic compounds with nitrogen hetero-atom(s) only. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:20.0%

Articles

Structure-activity relationship and site of binding of polyamine derivatives at the nicotinic acetylcholine receptor.

Eur. J. Biochem. 267(1) , 110-20, (2000)

Several wasp venoms contain philanthotoxins (PhTXs), natural polyamine amides, which act as noncompetitive inhibitors (NCIs) on the nicotinic acetylcholine receptor (nAChR). Effects of varying the str...

Liquid chromatographic methods for assay of carbamazepine, 10,11-dihydrocarbamazepine, and related compounds in carbamazepine drug substance and tablets.

J. Assoc. Off. Anal. Chem. 70(5) , 836-40, (1987)

Liquid chromatographic (LC) methods have been developed for the determination of carbamazepine, the impurity 10,11-dihydrocarbamazepine, and related compounds in carbamazepine drug substance and table...

An orthorhombic polymorph of 10,11-dihydrocarbamazepine.

Acta Crystallogr. C 62(Pt 5) , o240-2, (2006)

The title compound (systematic name: 10,11-dihydro-5H-dibenz[b,f]azepine-5-carboxamide), C15H14N2O, is shown to crystallize as an orthorhombic polymorph to complement the known monoclinic form. The mo...


More Articles


Related Compounds

  • cis-10,11-Dihydroxy-10,11-dihydrocarbamazepine
  • 10,11-trans-dihydroxy-10,11-dihydrocarbamazepine
  • 10,11,12-trihydroxyeicosatrienoic acid
  • 10,11-dihydro-4H-thieno[3,2-b][f]benzazepin-10-one
  • 10,11-dimethoxy-3-hydroxy-5,6,13,13a-tetrahydro-8H-dibenzo[a,g]quinolizine
  • 10,11-dihydro-5H-dibenzo[a,d][7]annulen-5-yl 4-nitrobenzoate
  • 4-((Cyclohexylamino)methyl)benzoic acid hydrochloride
  • 1-[(2,4-Dichlorophenyl)methyl]-N-(1,1-dimethylethyl)-2-methyl-1H-indole-3-methanamine
  • 2-Methoxy-6-(pyrazol-1-yl)-benzonitrile
  • 1H-3-Benzazepin-7-ol, 8-chloro-2,3,4,5-tetrahydro-5-(3-iodophenyl)-3-methyl-, (S)-
  • (2S)-4-(1-methyl-3-phenyl-1H-pyrazol-5-yl)butan-2-amine
  • 4-ethyl-1-[1-({[(9H-fluoren-9-yl)methoxy]carbonyl}amino)cyclopropaneamido]cyclohexane-1-carboxylic acid
  • (4-Methyl-tetrahydro-furan-2-yl)-methanol
  • N-(1-cyanocyclopentyl)-2-[4-(4-fluorobenzenesulfonyl)-1,4-diazepan-1-yl]acetamide
  • 4,5,6,7-Tetrahydrobenzo[d]isoxazole-3-carbaldehyde
  • tert-Butyl-DL-alanine