NECA

Suppliers

Names

[ CAS No. ]:
35920-39-9

[ Name ]:
NECA

[Synonym ]:
(2S,3S,4R,5R)-5-(6-Amino-9H-purin-9-yl)-N-ethyl-3,4-dihydroxytetrahydrofuran-2-carboxamide (non-preferred name)
(2S,3S,4R,5R)-5-(6-Amino-9H-purin-9-yl)-N-ethyl-3,4-dihydroxytetrahydro-2-furancarboxamide (non-preferred name)
5’-Ethylcarboxamido Adenosine
MFCD00069195
5'-Ethylcarboxamido Adenosine
1-(6-AMINO-9H-PURIN-9-YL)-1-DEOXY-N-ETHYL-β-D-RIBOFURANURONAMIDE
β-D-Ribofuranuronamide, 1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-
5'-(N-Ethylcarboxamido)adenosine
NECA

Chemical & Physical Properties

[ Density]:
1.9±0.1 g/cm3

[ Melting Point ]:
229-231ºC

[ Molecular Formula ]:
C12H16N6O4

[ Molecular Weight ]:
308.293

[ Exact Mass ]:
308.123291

[ PSA ]:
148.41000

[ LogP ]:
-0.48

[ Index of Refraction ]:
1.829

[ Water Solubility ]:
45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: 0.2 mg/mL Solutions may be stored for several days at 4?#x00b0;C.

MSDS

Toxicological Information

CHEMICAL IDENTIFICATION

RTECS NUMBER :
VJ2232000
CHEMICAL NAME :
Ribofuranuronamide, 1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-, hemihydrate
CAS REGISTRY NUMBER :
35920-39-9
LAST UPDATED :
199512
DATA ITEMS CITED :
2
MOLECULAR FORMULA :
C12-H16-N6-O4.1/2H2-O
MOLECULAR WEIGHT :
317.35
WISWESSER LINE NOTATION :
T56 BN DN FN HNJ IZ D- BT5OTJ CQ DQ EVM2 &QH 1/2

HEALTH HAZARD DATA

ACUTE TOXICITY DATA

TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Oral
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
5 mg/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
JMCMAR Journal of Medicinal Chemistry. (American Chemical Soc., Distribution Office Dept. 223, POB POB 57136, West End Stn., Washington, DC 20037) V.6- 1963- Volume(issue)/page/year: 23,313,1980
TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Intraperitoneal
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
500 ug/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
JMCMAR Journal of Medicinal Chemistry. (American Chemical Soc., Distribution Office Dept. 223, POB POB 57136, West End Stn., Washington, DC 20037) V.6- 1963- Volume(issue)/page/year: 23,313,1980

Safety Information

[ Symbol ]:

GHS06

[ Signal Word ]:
Danger

[ Hazard Statements ]:
H300

[ Precautionary Statements ]:
P264-P301 + P310

[ Personal Protective Equipment ]:
Eyeshields;Faceshields;full-face particle respirator type N100 (US);Gloves;respirator cartridge type N100 (US);type P1 (EN143) respirator filter;type P3 (EN 143) respirator cartridges

[ Hazard Codes ]:
T+: Very toxic;

[ Risk Phrases ]:
R28

[ Safety Phrases ]:
22-26-36-45

[ RIDADR ]:
UN 2811 6.1/PG 2

[ WGK Germany ]:
3

[ RTECS ]:
VJ2232000

[ Packaging Group ]:
I

[ Hazard Class ]:
6.1(a)

[ HS Code ]:
2934999090

Precursor & DownStream

Precursor

  • 5'-Ethylcarboxamido-2',3'-isopropylidene Adenosine
  • b-D-Ribofuranuronic acid,1-(6-amino-9H-purin-9-yl)-1-deoxy-2,3-O-(1-methylethylidene)-
  • Ethylamine
  • ethyl adenosine-5'-carboxylate
  • 2',3'-O-Isopropylideneadenosine
  • b-D-Ribofuranuronic acid,1-(6-amino-9H-purin-9-yl)-1-deoxy-
  • adenosine-5'-carboxylic acid 2-chloroethyl ester

DownStream

  • (2S,3S,4R,5R)-N-ethyl-3,4-dihydroxy-5-(1-hydroxy-6-imino-purin-9-yl)ox olane-2-carboxamide

Customs

[ HS Code ]: 2934999090

[ Summary ]:
2934999090. other heterocyclic compounds. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:20.0%

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Related Compounds

  • NECA
  • Dineca
  • b-neca
  • Dansyl-NECA
  • 2 inverted exclamation mark,3 inverted exclamation mark-O-isopropylidene-NECA
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  • 8-Fluoro-5-methyl-1,2,3,4-tetrahydroquinoline
  • 8-((Perfluoropropyl)thio)quinoline trifluoromethanesulfonate
  • {3-[(3-Aminopropyl)amino]propyl}(benzyl)amine
  • Phosphine oxide, hexylmethylphenyl-, (R)-