1,2,3,4-tetrahydro-6,7-dimethoxy-2-methyl-1-[2-(4-nitrophenyl)ethyl]-

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Names

[ CAS No. ]:
63937-57-5

[ Name ]:
1,2,3,4-tetrahydro-6,7-dimethoxy-2-methyl-1-[2-(4-nitrophenyl)ethyl]-

[Synonym ]:
4'-Nitromethopholine
Isoquinoline, 1,2,3,4-tetrahydro-6,7-dimethoxy-2-methyl-1-[2-(4-nitrophenyl)ethyl]-
6,7-Dimethoxy-2-methyl-1-[2-(4-nitrophenyl)ethyl]-1,2,3,4-tetrahydroisoquinoline
UNII:86JU2L138Q
1,2,3,4-tetrahydro-6,7-dimethoxy-2-methyl-1-[2-(4-nitrophenyl)ethyl]-

Chemical & Physical Properties

[ Density]:
1.2±0.1 g/cm3

[ Boiling Point ]:
496.2±45.0 °C at 760 mmHg

[ Melting Point ]:
91-92ºC

[ Molecular Formula ]:
C20H24N2O4

[ Molecular Weight ]:
356.416

[ Flash Point ]:
253.9±28.7 °C

[ Exact Mass ]:
356.173615

[ PSA ]:
67.52000

[ LogP ]:
4.08

[ Vapour Pressure ]:
0.0±1.3 mmHg at 25°C

[ Index of Refraction ]:
1.571

Toxicological Information

CHEMICAL IDENTIFICATION

RTECS NUMBER :
NX5035000
CHEMICAL NAME :
Isoquinoline, 1,2,3,4-tetrahydro-6,7-dimethoxy-2-methyl-1-(4-nitrop henethyl)-
CAS REGISTRY NUMBER :
63937-57-5
BEILSTEIN REFERENCE NO. :
1556086
LAST UPDATED :
199612
DATA ITEMS CITED :
1
MOLECULAR FORMULA :
C20-H24-N2-O4
MOLECULAR WEIGHT :
356.46
WISWESSER LINE NOTATION :
T66 CNT&J B2R DNW& C1 HO1 IO1

HEALTH HAZARD DATA

ACUTE TOXICITY DATA

TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Intravenous
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
10 mg/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
MDCHAG Medicinal Chemistry: A Series of Monographs. (Academic Press, Inc., 1 E. First St., Duluth, MN 55802) V.1- 1963- Volume(issue)/page/year: 5,290,1965

Safety Information

[ HS Code ]:
2933499090

Customs

[ HS Code ]: 2933499090

[ Summary ]:
2933499090. other compounds containing in the structure a quinoline or isoquinoline ring-system (whether or not hydrogenated), not further fused. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:20.0%


Related Compounds

  • rac-1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl (1R,2S)-2-(1H-1,2,4-triazol-3-yl)cyclopropane-1-carboxylate
  • tert-butyl (2S)-2-{3-[(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)oxy]-3-oxopropyl}-2-methylpyrrolidine-1-carboxylate
  • 1-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl) 4-ethyl 2-oxabicyclo[2.1.1]hexane-1,4-dicarboxylate
  • rac-1-tert-butyl 2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl) (2R,4S)-4-ethylpiperidine-1,2-dicarboxylate
  • 1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl 2-[4-chloro-2-(dimethylsulfamoyl)phenoxy]propanoate
  • 1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl (3S)-3-[3-(trifluoromethoxy)phenyl]butanoate
  • 1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl 1-cyclobutyl-2,2-difluorocyclopropane-1-carboxylate
  • rac-1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl (1R,2R)-2-(2-chloro-6-methoxyphenyl)cyclopropane-1-carboxylate
  • 1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl (1s,3s)-3-(tert-butoxy)cyclobutane-1-carboxylate
  • rac-1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl (1R,2S)-2-(4-fluorophenyl)cyclopentane-1-carboxylate
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