Molindone

Suppliers

Names

[ CAS No. ]:
7416-34-4

[ Name ]:
Molindone

[Synonym ]:
3-ethyl-2-methyl-5-morpholin-4-ylmethyl-1,5,6,7-tetrahydro-indol-4-one
MOLINDONE
molidone hydrochloride
EN-1733A

Chemical & Physical Properties

[ Density]:
1.14 g/cm3

[ Boiling Point ]:
462.9ºC at 760 mmHg

[ Melting Point ]:
180 - 181ºC

[ Molecular Formula ]:
C16H24N2O2

[ Molecular Weight ]:
276.37400

[ Flash Point ]:
233.7ºC

[ Exact Mass ]:
276.18400

[ PSA ]:
45.33000

[ LogP ]:
1.90070

[ Index of Refraction ]:
1.559

[ Water Solubility ]:
H2O: 19 mg/mL

Toxicological Information

CHEMICAL IDENTIFICATION

RTECS NUMBER :
NM3300000
CHEMICAL NAME :
Indol-4(5H)-one, 3-ethyl-6,7-dihydro-2-methyl-5-(morpholinomethyl)-
CAS REGISTRY NUMBER :
7416-34-4
LAST UPDATED :
199801
DATA ITEMS CITED :
2
MOLECULAR FORMULA :
C16-H24-N2-O2
MOLECULAR WEIGHT :
276.42
WISWESSER LINE NOTATION :
T56 BM FV&TJ C1 D2 G1- AT6N DOTJ

HEALTH HAZARD DATA

ACUTE TOXICITY DATA

TYPE OF TEST :
TDLo - Lowest published toxic dose
ROUTE OF EXPOSURE :
Oral
SPECIES OBSERVED :
Human
DOSE/DURATION :
714 ug/kg/D
TOXIC EFFECTS :
Behavioral - somnolence (general depressed activity) Behavioral - tremor Behavioral - antipsychotic
REFERENCE :
34ZIAG "Toxicology of Drugs and Chemicals," Deichmann, W.B., New York, Academic Press, Inc., 1969 Volume(issue)/page/year: -,402,1969
TYPE OF TEST :
TDLo - Lowest published toxic dose
ROUTE OF EXPOSURE :
Oral
SPECIES OBSERVED :
Human - man
DOSE/DURATION :
4285 ug/kg/3D-I
TOXIC EFFECTS :
Behavioral - muscle weakness Lungs, Thorax, or Respiration - cyanosis Kidney, Ureter, Bladder - changes in tubules (including acute renal failure, acute tubular necrosis)
REFERENCE :
JCLPDE Journal of Clinical Psychiatry. (Physicians Postgraduate Press, Inc., POB 240008, Memphis, TN 38124) V.39- 1978- Volume(issue)/page/year: 47,607,1986

Safety Information

[ Hazard Codes ]:
Xn: Harmful;

[ Risk Phrases ]:
22

[ RIDADR ]:
UN 2811 6.1/PG 3

[ WGK Germany ]:
3

[ RTECS ]:
NM3325000

Synthetic Route

Precursor & DownStream

Precursor

  • 4,4'-Methylenedimorpholine
  • 2-Methyl-3-ethyl-4-oxo-4,5,6,7-tetrahydroindole
  • 2-Hydroxyimino-3-pentanone
  • 1,3-Cyclohexanedione
  • 2,3-Pentanedione

DownStream


Related Compounds

  • Molindone-d8
  • Molindone hydrochloride
  • 4-((Cyclohexylamino)methyl)benzoic acid hydrochloride
  • 1-[(2,4-Dichlorophenyl)methyl]-N-(1,1-dimethylethyl)-2-methyl-1H-indole-3-methanamine
  • 2-Methoxy-6-(pyrazol-1-yl)-benzonitrile
  • 1H-3-Benzazepin-7-ol, 8-chloro-2,3,4,5-tetrahydro-5-(3-iodophenyl)-3-methyl-, (S)-
  • (4-Methyl-tetrahydro-furan-2-yl)-methanol
  • N-(1-cyanocyclopentyl)-2-[4-(4-fluorobenzenesulfonyl)-1,4-diazepan-1-yl]acetamide
  • 4,5,6,7-Tetrahydrobenzo[d]isoxazole-3-carbaldehyde
  • tert-Butyl-DL-alanine
  • 4-amino-N-[2-tert-butyl-1-(tetrahydro-2H-pyran-4-ylmethyl)-1H-benzimidazol-5-yl]-N-ethylbenzenesulfonamide
  • 5-(3-chloro-1H-pyrazol-1-yl)-2-(chlorodifluoromethyl)pyrimidine