Methiothepin mesylate

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Names

[ Name ]:
Methiothepin mesylate

[Synonym ]:
Methiothepin mesylate salt
Methiothepin methanesulfonate
Methiothepin mesylate
Metitepine mesylate salt
Piperazine,1-(10,11-dihydro-8-(methylthio)dibenzo(b,f)thiepin-10-yl)-4-methyl-,methanesulfonate
1-[10,11-Dihydro-8-(methylthio)dibenzo[b,f]thiepin-10-yl]-4-methylpiperazine mesylate salt

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₁H₂₈N₂O₃S₃

[ Molecular Weight ]:
452.65400

[ Exact Mass ]:
452.12600

[ PSA ]:
119.83000

[ LogP ]:
4.86490

[ Storage condition ]:
2-8℃

MSDS

Click to get detail MSDS

Safety Information

[ Personal Protective Equipment ]:
Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter

[ RIDADR ]:
NONH for all modes of transport

Articles

Characterization of the commercially-available fluorescent chloroquine-BODIPY conjugate, LynxTag-CQGREEN, as a marker for chloroquine resistance and uptake in a 96-well plate assay.

PLoS ONE 9(10) , e110800, (2014)

Chloroquine was a cheap, extremely effective drug against Plasmodium falciparum until resistance arose. One approach to reversing resistance is the inhibition of chloroquine efflux from its site of ac...

Functional, endogenously expressed 5-hydroxytryptamine 5-ht7 receptors in human vascular smooth muscle cells.

Br. J. Pharmacol. 117 , 993-994, (1996)

Human uterine artery smooth muscle cells in culture were shown to express constitutively both 5-ht7 receptor mRNA and 5-ht7-like receptors functionally linked to cyclic AMP formation. 5-Carboxamidotry...

Characterisation of 5-HT receptors in human coronary arteries by molecular and pharmacological techniques.

Eur. J. Pharmacol. 372 , 49-56, (1999)

5-Hydroxytryptamine (5-HT) can produce both vasoconstrictor and vasorelaxant effects in human coronary arteries and the response to 5-HT can be influenced by the presence of disease. The aim of the pr...