Raloxifene HCl

Suppliers

Names

[ Name ]:
Raloxifene HCl

[Synonym ]:
[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophen-3-yl][4-(2-piperidin-1-ylethoxy)phenyl]methanone hydrochloride
[6-Hydroxy-2-(4-hydroxyphenyl)-1-benzothiophen-3-yl]{4-[2-(piperidin-1-yl)ethoxy]phenyl}methanone hydrochloride (1:1)
Raloxifene HCl
[6-Hydroxy-2-(4-hydroxyphenyl)-1-benzothiophen-3-yl][4-(2-piperidin-1-ylethoxy)phenyl]methanonhydrochlorid
1-[2-(4-{[6-Hydroxy-2-(4-hydroxyphenyl)-1-benzothiophen-3-yl]carbonyl}phenoxy)ethyl]piperidinium chloride
[6-Hydroxy-2-(4-hydroxyphenyl)-1-benzothiophen-3-yl]{4-[2-(1-piperidinyl)ethoxy]phenyl}methanone hydrochloride (1:1)
Methanone, [6-hydroxy-2-(4-hydroxyphenyl)benzo[b]thien-3-yl][4-[2-(1-piperidinyl)ethoxy]phenyl]-, hydrochloride (1:1)
methanone, [6-hydroxy-2-(4-hydroxyphenyl)benzo[b]thien-3-yl][4-[2-(1-piperidinyl)ethoxy]phenyl]-, hydrochloride
6-Hydroxy-2-(p-hydroxyphenyl)benzo(b)thien-3-yl-p-(2-piperidinoethoxy)phenyl ketone hydrochloride
MFCD01938233
Raloxifene hydrochloride
Raloxifene (hydrochloride)

Chemical & Physical Properties

[ Density]:
1.285g/cm3

[ Boiling Point ]:
728.2ºC at 760 mmHg

[ Melting Point ]:
143-147ºC

[ Molecular Formula ]:
C₂₈H₂₈ClNO₄S

[ Molecular Weight ]:
510.044

[ Flash Point ]:
394.2ºC

[ Exact Mass ]:
509.142761

[ PSA ]:
98.24000

[ LogP ]:
6.81510

[ Index of Refraction ]:
1.654

[ Storage condition ]:
-20°C Freezer

[ Water Solubility ]:
DMSO: 28 mg/mL, soluble

Safety Information

[ Personal Protective Equipment ]:
Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter

[ Hazard Codes ]:
Xi

[ Risk Phrases ]:
R36/37/38

[ Safety Phrases ]:
22-24/25

[ RIDADR ]:
NONH for all modes of transport

[ WGK Germany ]:
3

Synthetic Route

Click to get detail synthetic route

Precursor & DownStream

Precursor

[4-(6-acetyloxy-1-benzothiophen-2-yl)phenyl] acetate
4-[2-(1-Pipiridine)ethoxybenzoic acid hydrochloride
Raloxifene Bismethyl Ether hydrochloride
6-Methoxy-2-(4-methoxyphenyl)-1-benzothiophene
[6-[(methylsulfonyl)oxy]-2-[4-[(methylsulfonyl)oxy]phenyl]benzo[b]thien-3-yl][4-[2-(1-pyrrolidinyl)ethoxy]phenyl]methanone hydrochloride
Raloxifene
4-Methoxythiophenol
4-(2-PIPERIDINOETHOXY)BENZOIC ACID HYDROCHLORIDE
4-Methoxy-alpha-[(3-methoxyphenyl)thio]acetophenone
PTP inhibitor 1

DownStream

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