Deoxycholic acid

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Names

[ CAS No. ]:
83-44-3

[ Name ]:
Deoxycholic acid

[Synonym ]:
7-DEOXYCHOLIC ACID
Cholan-24-oic acid, 3,12-dihydroxy-, (3α,5β,12α)-
5b-Deoxycholic acid
Deoxycholatic acid
EINECS 201-478-5
Deoxycholic acid
17b-(1-Methyl-3-carboxypropyl)etiocholane-3a,12a-diol
deoxy-Cholic acid
(3α,5β,12α)-3,12-Dihydroxycholan-24-oic acid
7α-Deoxycholic acid
Kybella
3α,12α-dihydroxy-5β-cholan-24-oic acid
ATX-101
5b-Cholanic acid-3a,12a-diol
Dihydroxycholanoic acid
Cholic acid, deoxy-
(3a,5b,12a)-3,12-Dihydroxy-5-cholan-24-oic Acid
(4R)-4-[(3R,5R,8R,9S,10S,12S,13R,14S,17R)-3,12-Dihydroxy-10,13-dimethylhexadecahydro-1H-cyclopenta[a]phenanthren-17-yl]pentanoic acid
MFCD00003673

Chemical & Physical Properties

[ Density]:
1.1±0.1 g/cm3

[ Boiling Point ]:
547.1±35.0 °C at 760 mmHg

[ Melting Point ]:
171-174 °C(lit.)

[ Molecular Formula ]:
C24H40O4

[ Molecular Weight ]:
392.572

[ Flash Point ]:
298.8±22.4 °C

[ Exact Mass ]:
392.292664

[ PSA ]:
77.76000

[ LogP ]:
4.66

[ Vapour Pressure ]:
0.0±3.3 mmHg at 25°C

[ Index of Refraction ]:
1.543

[ Water Solubility ]:
0.24 g/L (15 ºC)

MSDS

Toxicological Information

CHEMICAL IDENTIFICATION

RTECS NUMBER :
FZ2100000
CHEMICAL NAME :
5-beta-Cholan-24-oic acid, 3-alpha,12-alpha-dihydroxy-
CAS REGISTRY NUMBER :
83-44-3
BEILSTEIN REFERENCE NO. :
3219882
LAST UPDATED :
199701
DATA ITEMS CITED :
15
MOLECULAR FORMULA :
C24-H40-O4
MOLECULAR WEIGHT :
392.64
WISWESSER LINE NOTATION :
L E5 B666TJ A1 DQ E1 FY1&2VQ OQ

HEALTH HAZARD DATA

ACUTE TOXICITY DATA

TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Oral
SPECIES OBSERVED :
Rodent - rat
DOSE/DURATION :
1 gm/kg
TOXIC EFFECTS :
Behavioral - food intake (animal) Nutritional and Gross Metabolic - weight loss or decreased weight gain
TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Oral
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
1 gm/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Intravenous
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
130 mg/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
TYPE OF TEST :
LDLo - Lowest published lethal dose
ROUTE OF EXPOSURE :
Intravenous
SPECIES OBSERVED :
Rodent - rabbit
DOSE/DURATION :
2 gm/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
TYPE OF TEST :
TDLo - Lowest published toxic dose
ROUTE OF EXPOSURE :
Administration onto the skin
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
2700 mg/kg/10W-I
TOXIC EFFECTS :
Tumorigenic - equivocal tumorigenic agent by RTECS criteria Skin and Appendages - tumors
TYPE OF TEST :
TDLo - Lowest published toxic dose
ROUTE OF EXPOSURE :
Subcutaneous
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
1120 mg/kg/22W-I
TOXIC EFFECTS :
Tumorigenic - equivocal tumorigenic agent by RTECS criteria Tumorigenic - tumors at site of application
TYPE OF TEST :
TD - Toxic dose (other than lowest)
ROUTE OF EXPOSURE :
Subcutaneous
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
1400 mg/kg/22W-I
TOXIC EFFECTS :
Tumorigenic - equivocal tumorigenic agent by RTECS criteria Tumorigenic - tumors at site of application
TYPE OF TEST :
TDLo - Lowest published toxic dose
ROUTE OF EXPOSURE :
Intraperitoneal
DOSE :
166 mg/kg
SEX/DURATION :
female 12-19 day(s) after conception
TOXIC EFFECTS :
Reproductive - Fertility - post-implantation mortality (e.g. dead and/or resorbed implants per total number of implants) Reproductive - Effects on Embryo or Fetus - fetotoxicity (except death, e.g., stunted fetus)

MUTATION DATA

TYPE OF TEST :
Morphological transformation
TEST SYSTEM :
Rodent - hamster Embryo
DOSE/DURATION :
7250 ug/L
REFERENCE :
TOLED5 Toxicology Letters. (Elsevier Science Pub. B.V., POB 211, 1000 AE Amsterdam, Netherlands) V.1- 1977- Volume(issue)/page/year: 9,177,1981 *** NIOSH STANDARDS DEVELOPMENT AND SURVEILLANCE DATA *** NIOSH OCCUPATIONAL EXPOSURE SURVEY DATA : NOHS - National Occupational Hazard Survey (1974) NOHS Hazard Code - 80398 No. of Facilities: 153 (estimated) No. of Industries: 2 No. of Occupations: 7 No. of Employees: 3527 (estimated) NOES - National Occupational Exposure Survey (1983) NOES Hazard Code - 80398 No. of Facilities: 82 (estimated) No. of Industries: 2 No. of Occupations: 5 No. of Employees: 2416 (estimated) No. of Female Employees: 1577 (estimated)

Safety Information

[ Symbol ]:

GHS07

[ Signal Word ]:
Warning

[ Hazard Statements ]:
H302

[ Precautionary Statements ]:
P301 + P312 + P330

[ Personal Protective Equipment ]:
dust mask type N95 (US);Eyeshields;Gloves

[ Hazard Codes ]:
Xn:Harmful

[ Risk Phrases ]:
R22;R36/37/38

[ Safety Phrases ]:
S26-S36-S37/39

[ RIDADR ]:
NONH for all modes of transport

[ WGK Germany ]:
3

[ RTECS ]:
FZ2100000

Synthetic Route

Precursor & DownStream

Precursor

  • Cholan-24-oic acid,3,12-dihydroxy-, methyl ester, (3a,5b,12a)-
  • Methyl 3α-hydroxy-12-oxo-5β-cholan-24-oate
  • 5BETA-CHOLANIC ACID-3ALPHA,12ALPHA-DIOL 3-ACETATE METHYL ESTER
  • Lithocholic acid
  • 5.beta.-Chol-9 (11)-en-24-oic acid, 3.alpha.-hydroxy-12-oxo-, methyl ester, acetate
  • 9-Hydroxyandrost-4-ene-3,17-dione
  • 9alpha-hydroxy-5beta-androstane-3,17-dione
  • 5β-androst-9(11)-ene-3,17-dione
  • 9(11), (5-BETA)-ANDROSTEN-3-ALPHA-OL-17-ONE

DownStream

  • GLYCODEOXYCHOLIC ACID
  • Cholan-24-oic acid,3,12-dihydroxy-, methyl ester, (3a,5b,12a)-
  • 5b-Cholan-24-oic acid, 3a,12b-dihydroxy-11-oxo- (8CI)
  • Lithocholic acid
  • (S)-(+)-2-Aminobutane
  • Cholan-24-oic acid,3,12-bis(formyloxy)-, (3a,5b,12a)-
  • 1,3-Dicyclohexylurea
  • taurodeoxycholic acid

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Related Compounds

  • deoxycholic acid
  • deoxycholic acid
  • deoxycholic acid
  • 3-deoxycholic acid
  • Deoxycholic acid-d4
  • Deoxycholic Acid-d5
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