Journal of Organic Chemistry 2008-08-15

Copper-mediated N-cyclopropylation of azoles, amides, and sulfonamides by cyclopropylboronic acid.

Sébastien Bénard, Luc Neuville, Jieping Zhu

文献索引：J. Org. Chem. 73 , 6441, (2008)

全文：HTML全文

摘要

Reaction of azoles, amides, and sulfonamides in dichloroethane with readily available cyclopropylboronic acid in the presence of copper acetate and sodium carbonate afforded the N-cyclopropyl derivatives in good to excellent yields.

相关化合物

  • 环丙基硼酸

相关文献：

Palladium-catalyzed decarboxylative coupling of isatoic anhydrides with arylboronic acids.

2011-11-18

[Org. Lett. 13 , 6114-6117, (2011)]

Palladium-catalyzed alkylation of sp2 and sp3 C-H bonds with methylboroxine and alkylboronic acids: two distinct C-H activation pathways.

2006-10-04

[J. Am. Chem. Soc. 128 , 12634, (2006)]

2-(2-Aminothiazol-4-yl)pyrrolidine-based tartrate diamides as potent, selective and orally bioavailable TACE inhibitors.

2011-05-15

[Bioorg. Med. Chem. Lett. 10th ed., 21 , 3172-3176, (2011)]

[Tetrahedron Lett. 43 , 6987-6990, (2002)]

Microwave-assisted N-cyclopropylation of pyridinols with cyclopropyl boronic acid Tambe, Y. B.; et al.

[Synth. Commun. 9th ed., 42 , 1341-1348, (2012)]

更多文献...