Journal of Organic Chemistry 2006-10-13

Molecular iodine-catalyzed facile procedure for N-Boc protection of amines.

Ravi Varala, Sreelatha Nuvula, Srinivas R Adapa

文献索引：J. Org. Chem. 71 , 8283, (2006)

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摘要

An efficient and practical protocol for the protection of various structurally and electronically divergent aryl and aliphatic amines using (Boc)2O in the presence of a catalytic amount of molecular iodine (10 mol %) under solvent-free conditions at ambient temperature is presented.

相关化合物

  • 1-Boc-哌嗪

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