Journal of Organic Chemistry 2007-05-11

Reactions of nitroso hetero-Diels-Alder cycloadducts with azides: stereoselective formation of triazolines and aziridines.

Brian S Bodnar, Marvin J Miller

文献索引：J. Org. Chem. 72 , 3929, (2007)

全文：HTML全文

摘要

The addition of azides to acylnitroso hetero-Diels-Alder cycloadducts derived from cyclopentadiene affords exo-triazolines in excellent yield. The reaction is greatly affected by the level of alkene strain, while sterically demanding azides do not hinder the reaction. Conversion of the triazolines to aziridines is also described.

相关化合物

  • N-叔丁氧羰基羟胺

相关文献：

N-O chemistry for antibiotics: discovery of N-alkyl-N-(pyridin-2-yl)hydroxylamine scaffolds as selective antibacterial agents using nitroso Diels-Alder and ene chemistry.

2011-10-13

[J. Med. Chem. 54 , 6843-58, (2011)]

Prodrugs of nitroxyl as inhibitors of aldehyde dehydrogenase.

1992-10-02

[J. Med. Chem. 35 , 3648, (1992)]

D.S. Jones et al.

[Tetrahedron Lett. 41 , 1531, (2000)]

M. Adamczyk, R.E. Reddy

[Synth. Commun. 31 , 579, (2001)]

J.M. Altenburger et al.

[Tetrahedron Lett. 33 , 5055, (1992)]

更多文献...