α-甲基血清素 马来酸盐

α-methyl Serotonin (maleate) is an agonist of serotonin (5-HT) receptors. It binds selectively to 5-HT1A, 5-HT1B, 5-HT1C, and 5-HT1D receptors over 5-HT1E receptors. It is also selective for 5-HT2B and 5-HT2C receptors over 5-HT2A receptors. α-methyl Serotonin potentiates motor neuron depolarizations induced by NMDA in the presence of the NMDA receptor antagonist memantine. It also increases dopamine release in a dose-dependent manner. α-methyl Serotonin increases systolic blood pressure and transiently increases heart rate.

[ 熔点 ]:
191 - 193 °C

[ 分子式 ]:
C₁₅H₁₈N₂O₅

[ 分子量 ]:
306.31400

[ 精确质量 ]:
306.12200

[ PSA ]:
136.64000

[ LogP ]:
2.17530

[ 外观性状 ]:
白色米色粉末

[ 储存条件 ]:
20°C

详细MSDS(安全技术说明书)

[ 个人防护装备 ]:
Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter

[ 危险品运输编码 ]:
NONH for all modes of transport

[ 海关编码 ]:
2933990090

[ 海关编码 ]: 2933990090

[ 中文概述 ]:
2933990090. 其他仅含氮杂原子的杂环化合物. 增值税率:17.0%. 退税率:13.0%. 监管条件:无. 最惠国关税:6.5%. 普通关税:20.0%

[ 申报要素 ]: 品名, 成分含量, 用途, 乌洛托品请注明外观, 6－己内酰胺请注明外观, 签约日期

[ Summary ]:
2933990090. heterocyclic compounds with nitrogen hetero-atom(s) only. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:20.0%

5-HT1 and 5-HT2 binding profiles of the serotonergic agents alpha-methylserotonin and 2-methylserotonin.

J. Med. Chem. 33 , 755-758, (1990)

alpha-Methyl-5-hydroxytryptamine (alpha-Me-5-HT; 2) and 2-methyl-5-hydroxytryptamine (2-Me-5-HT; 3) are considered to be 5-HT2-selective and 5-HT3-selective agents, respectively. These agents were syn...

Serotonin via 5-HT1B and 5-HT2B receptors stimulates anion secretion in the rat epididymal epithelium.

J. Physiol. 519 , 519, (1999)

1. The short-circuit current (Isc) technique was used to study the role of 5-hydroxytryptamine (5-HT) in the regulation of anion secretion in cultured rat cauda epididymal epithelia. 2. 5-HT, the 5-HT...

Effects of serotonin-1 and serotonin-2 receptor agonists on neuronal activity in the nucleus tractus solitarius.

J. Auton. Nerv. Syst. 56 , 119-124, (1995)

Spontaneous neuronal activity in the solitary tract nucleus was recorded extracellularly in a brain slice preparation during bath-application of 5-HT1 and 5-HT2 receptor-selective agonists and antagon...

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公司名：上海化源世纪贸易有限公司

区域：上海市普陀区

价格：

联系人：徐经理

产品详情：α-甲基血清素 马来酸盐

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公司名：上海脉铂医药科技有限公司

区域：上海市嘉定区

价格：
￥8789.0/50mg ￥2069.0/10mg ￥需询单/1g ￥需询单/1g

联系人：李先生

产品详情：α-Methyl-5-hydroxytryptamine maleate

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公司名：上海创赛科技有限公司

区域：上海市嘉定区

价格：
￥8624.0/50mg ￥2038.4/10mg

联系人：夏言

产品详情：α-Methyl-5-hydroxytryptamine maleate

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公司名：上海阿拉丁生化科技股份有限公司

区域：上海市浦东新区

价格：
￥1500.0/50mg ￥390.0/100mg ￥需询单/1g ￥需询单/1g

联系人：阿拉丁

产品详情：5-羟色胺马来酸α-甲酯

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