11-(1-甲基哌啶-4-亚基)-6,11-二氢-5H-苯并[5,6]环庚[1,2-b]吡啶二马来酸盐

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发布时间： 2024-07-15 12:35:08

CAS号：3978-86-7

常用名： 马来酸阿扎他啶

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纯度： 98.0%

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用途： Azatadine dimaleate is an histamine and cholinergic inhibitor with IC50 of 6.5 nM and 10 nM, respectively.Target: Histamine ReceptorAzatadine, a new antihistamine, was evaluated for its efficacy in 20 patients with chronic allergic rhinitis. Eighty percent of patients had symptomatic relief with a twice daily dosage of 2 mg. Sedation was volunteered as a side effect by six of the patients and was admitted by two further patients after specific questioning. A choice reaction time test gave slowing of motor function in these sedated patients. Four of the previously sedated patients experienced good symptomatic control with minimal sedation when the azatadine dose was reduced to 1 mg twice daily; slowing of motor function was not observed at this, the normal recommended dose.Azatadine delays the onset of dyspnea-induced by aerosolized histamine, acetylcholine and serotonin in the conscious guinea-pig with PD50 of 0.01 mg/kg, 0.739 mg/kg and 0.86 mg/kg. Azatadine protects conscious guinea-pigs against death induced by the intravenous injection of histamine with oral PD50 of 0.009 mg/kg in guinea-pig and 0.22 mg/kg in mice. 物理化学性质： CAS号：3978-86-7 常用中文名：马来酸阿扎他啶常用英文名：Azatadine dimaleate 分子式：C28H30N2O8 分子量：522.546 密度：N/A 沸点：450.1ºC at 760 mmHg 熔点：152-154° 闪点：226ºC 储存条件：室温，干燥

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公司名：上海念兴实业有限公司推荐

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2022-02-19 价格：￥60.9 Azatadine dimaleate

2021-02-06 价格：￥2149.0 Azatadine dimaleate

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马来酸阿扎他啶价格

11-(1-甲基哌啶-4-亚基)-6,11-二氢-5H-苯并[5,6]环庚[1,2-b]吡啶二马来酸盐

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