Non-imidazole heterocyclic histamine H 3 receptor antagonists

W Chai, JG Breitenbucher, A Kwok, X Li, V Wong…

文献索引：Chai, Wenying; Breitenbucher, J. Guy; Kwok, Annette; Li, Xiaobing; Wong, Victoria; Carruthers, Nicholas I.; Lovenberg, Timothy W.; Mazur, Curt; Wilson, Sandy J.; Axe, Frank U.; Jones, Todd K. Bioorganic and Medicinal Chemistry Letters, 2003 , vol. 13, # 10 p. 1767 - 1770

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被引用次数: 90

摘要

Continued exploration of the SAR around the lead imidazopyridine histamine H3 antagonist 1 has led to the discovery of several related series of heterocyclic histamine H3 antagonists. The synthesis and SAR of indolizine, indole and pyrazolopyridine based compounds are now described.