Benzothiophene inhibitors of MK2. Part 1: Structure–activity relationships, assessments of selectivity and cellular potency

DR Anderson, MJ Meyers, RG Kurumbail…

文献索引：Bioorganic and Medicinal Chemistry Letters, , vol. 19, # 16 p. 4878 - 4881

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被引用次数: 34

摘要

... Bioorganic & Medicinal Chemistry Letters. ... In summary, we have reported an additional chemical series of potent MK2 inhibitors with improved cellular potency and that the observed cellular potency is within the mechanism of action. ...