Abstract Synthesis of 5, 6-dimethoxyquinazolin-2 (1H)-one derivatives was the subject of investigations leading to the preparation of title compounds 11, 13, 14 and 26. Target quinazolines 1 were synthesized in three ways; the route starting from o-vanillin via the intermediacy of 6-amino-2, 3-dimethoxyacetophenone (19) was used for most of the preparative work. The unexpected formation of an acid-labile dimer of 13 was discovered ...
[Bandurco, Victor T.; Schwender, Charles F.; Bell, Stanley C.; Combs, Donald W.; Kanojia, Ramesh M.; et al. Journal of Medicinal Chemistry, 1987 , vol. 30, # 8 p. 1421 - 1426]
![Benzaldehyde,3-methoxy-2-[(phenylsulfonyl)oxy]结构式](https://image.chemsrc.com/caspic/344/2426-85-9.png)
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