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依克立达盐酸盐

更新时间:2025-08-30 15:40:25

常用名 依克立达盐酸盐 CAS号 143851-98-3
价格 ¥需询单/1mg 纯度 98.0%
备货期 3天 库存 现货
 产品详情(用途,包装等)
用途:
Elacridar Hcl (GF120918; GW0918) is a P-glycoprotein inhibitor, and has been used both in vitro and in vivo as a tool inhibitor of P-glycoprotein (Pgp) to investigate the role of transporters in the disposition of various test molecules.IC50 value:Target: P-glycoprotein In vitro, GF120918A demonstrated high plasma protein binding across species, although a definitive protein binding evaluation was precluded by poor recovery, particularly in buffer and in mouse, rat, and dog plasma. GF120918A did not demonstrate potent inhibition of several human cytochrome P450 enzymes evaluated in vitro, with IC(50) values well above concentrations anticipated to be achieved in vivo. Together, these data confirm the utility of GF120918A as a tool P-glycoprotein inhibitor in preclinical species and offer additional guidance on preclinical dose regimens likely to produce P-glycoprotein-mediated effects.
物理化学性质:
CAS号:143851-98-3
常用中文名:依克立达盐酸盐
常用英文名:Elacridar hydrochloride
分子式:C34H34ClN3O5
分子量:600.10400
密度:N/A
沸点:701.6ºC at 760 mmHg
熔点:N/A
闪点:378.1ºC
储存条件:2-8℃

供应商信息

上海泽涵生物医药科技有限公司

认证状态:未认证供应商
电话:021-61350663
地址:上海浦东新区丽正路1628号4幢4045室
地区: 上海市 上海市 浦东新区
联系人:薛经理
联系人电话:13052117465
邮件:sales@zehanbiopharma.com
网址:http://www.zehanbiopharma.com
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上海泽涵生物医药科技有限公司是集医药化学品(含中间体)、精细化学品和生物医药产品的研究、开发、生产、产品销售、技术服务于一体的高新企业。
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参考价格:$91/10mg
其他供应商价格:
2022-11-29 Elacridar hydrochloride
价格:¥需询单
2021-02-06 Elacridar hydrochloride
价格:¥1707.0
2022-02-19 Elacridar hydrochloride
价格:¥476.9
2018-10-30 依克立达盐酸盐
价格:¥需询单
2022-05-12 Elacridar HCl
价格:$需询单

查看所有价格,请点击依克立达盐酸盐价格