| 常用名 | EGF/FGF/PDGF受体酪氨酸激酶抑制剂 | CAS号 | 1135256-66-4 |
|---|---|---|---|
| 价格 | ¥1963.0/2mg ¥需询单/1g ¥需询单/1g ¥需询单/1g | 纯度 | 97.0% |
| 备货期 | 1天 | 库存 | 现货 |
| 产品网页 | http://www.aladdin-e.com/zh_cn/E337817.html | ||
| 产品详情(用途,包装等)
用途: EGF / FGF / PDGF受体酪氨酸激酶抑制剂是一种细胞可渗透且可逆的蛋白酪氨酸激酶抑制剂,可抑制人Flg(FGFR-1),PDGFR-β,c-Scr和EGFR,同时对InsR,PKC,或CDK4 / Cyclin D1。EGF / FGF / PDGF受体酪氨酸激酶抑制剂的抑制作用在c-Src情况下显示为非竞争性,在Flg(FGFR-1),PDGFR-β和EGFR情况下显示为ATP竞争性。 EGF/FGF/PDGF Receptor Tyrosine Kinase Inhibitor is a cell-permeable and reversible protein tyrosine kinase inhibitor that inhibits human Flg (FGFR-1), PDGFR-β, c-Scr, and EGFR, meanwhile exhibiting minimal activity against InsR, PKC, or CDK4/Cyclin D1. Inhibition by EGF/FGF/PDGF Receptor Tyrosine Kinase Inhibitor is shown to be noncompetitive in the case of c-Src, but ATP-competitive in the case of Flg (FGFR-1), PDGFR-β, and EGFR. 物理化学性质: CAS号:1135256-66-4 常用中文名:EGF/FGF/PDGF受体酪氨酸激酶抑制剂 常用英文名:EGF/FGF/PDGF receptor tyrosine kinase inhibitor 分子式:C18H18Cl2N6O 分子量:405.28 密度:~1.4 g/cm3(Predicted) 沸点:594.56° C (Predicted) 熔点:256.77° C (Predicted) 闪点:N/A 储存条件:2-8°C储存 |