| 常用名 | NGB 2904 hydrochloride | CAS号 | 189061-11-8 |
|---|---|---|---|
| 价格 | ¥8720.0/50mg ¥需询单/1g ¥需询单/1g ¥需询单/1g | 纯度 | 98.0% |
| 备货期 | 1天 | 库存 | 现货 |
| 产品网页 | http://www.aladdin-e.com/zh_cn/N287046.html | ||
| 产品详情(用途,包装等)
用途: NGB 2904 hydrochloride is a potent, selective, orally active and brain-penetrated antagonist of dopamine D3 receptor, with a Ki of 1.4 nM. NGB 2904 hydrochloride shows selectivity for D3 over D2, 5-HT2, α1, D4, D1 and D5 receptors (Kis=217, 223, 642, >5000, >10000 and >10000 nM, respectively). NGB 2904 hydrochloride antagonizes Quinpirole-stimulated mitogenesis. NGB 2904 hydrochloride can inhibit Cocaine's rewarding effects and Cocaine-induced reinstatement of drug-seeking behavior[1][2]. 物理化学性质: CAS号:189061-11-8 常用中文名:NGB 2904 hydrochloride 常用英文名:NGB 2904 hydrochloride 分子式:C28H30Cl3N3O 分子量:530.916 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A 储存条件:-20°C,密闭,干燥 |