| 常用名 | JTV-519 fumarate | CAS号 | 1883549-36-7 |
|---|---|---|---|
| 价格 | ¥需询单/1mg ¥需询单/1g ¥需询单/1g ¥需询单/1g | 纯度 | 98.0% |
| 备货期 | 1天 | 库存 | 现货 |
| 产品网页 | http://www.aladdin-e.com/zh_cn/J275634.html | ||
| 产品详情(用途,包装等)
用途: JTV-519 (K201) is a Ca2+-dependent blocker of SERCA and a partial agonist of ryanodine receptors (RyRs); displays Ca(2+)-dependent inhibition of SERCA-dependent ATPase activity with IC50 of 9 uM at 0.25 Ca2+ in cardiac muscle; may prevent abnormal Ca(2+) leak from the sarcoplasmic reticulum (SR) in the ischemic heart and skeletal muscle (SkM) by stabilizing the ryanodine receptors (RyRs; RyR1 and RyR2, respectively). Heart Arrhythmia Phase 2 Discontinued 物理化学性质: CAS号:1883549-36-7 常用中文名:JTV-519 fumarate 常用英文名:JTV-519 fumarate 分子式:C29H36N2O6S 分子量:540.675 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A |