| 常用名 | 咪唑斯汀 | CAS号 | 108612-45-9 |
|---|---|---|---|
| 价格 | ¥需询单/10mg ¥需询单/25mg ¥需询单/50mg ¥需询单/100mg | 纯度 | 99.9% |
| 备货期 | 需询单 | 库存 | 现货 |
| 产品详情(用途,包装等)
用途: Mizolastine is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions. Target: Histamine H1-receptorMizolastine is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions. It does not prevent the actual release of histamine from mast cells, just prevents it binding to receptors. Side effects can include dry mouth and throat.Mizolastine has demonstrated antiallergic effects in animals and healthy volunteers and anti-inflammatory activity in animal models. Double-blind trials have shown mizolastine to be significantly more effective than placebo and as effective as other second generation antihistamine agents, such as loratadine or cetirizine, in the management of patients with perennial or seasonal allergic rhinitis and in patients with chronic idiopathic urticaria. Available data also suggest that prophylactic administration of mizolastine is significantly more effective than placebo and as effective as prophylactic terfenadine in delaying the onset of symptoms of seasonal allergic rhinitis. 物理化学性质: CAS号:108612-45-9 常用中文名:咪唑斯汀 常用英文名:Mizolastine 分子式:C24H25FN6O 分子量:432.493 密度:1.3±0.1 g/cm3 沸点:N/A 熔点:217° 闪点:N/A 储存条件:室温 |